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CAS RN: 199739-10-1 | Product Number: P2967
Paliperidone Palmitate
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Purity: >98.0%(T)(HPLC)
Synonyms:
- 9-Hydroxyrisperidone Palmitate
- 3-[2-[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]ethyl]-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl Palmitate
Product Documents:
| Size | Unit Price | Same Day | 2-3 Business Days | Other Lead Time |
Shipping Information
|
|---|---|---|---|---|---|
| 100MG |
$62.00
|
10 | 0 | Contact Us | |
| 1G |
$362.00
|
4 | 12 | Contact Us |
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* The storage conditions are subject to change without notice.
| Product Number | P2967 |
| Purity / Analysis Method | >98.0%(T)(HPLC) |
| Molecular Formula / Molecular Weight | C__3__9H__5__7FN__4O__4 = 664.91 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature | Refrigerated (0-10°C) |
| Store Under Inert Gas | Store under inert gas |
| Condition to Avoid | Air Sensitive,Heat Sensitive |
| Packaging and Container | 100MG-Glass Bottle with Plastic Insert (View image), 1G-Glass Bottle with Plastic Insert (View image) |
| CAS RN | 199739-10-1 |
| Reaxys Registry Number | 15026585 |
| MDL Number | MFCD24386477 |
Specifications
| Appearance | White to Light yellow powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| Purity(Volumetric Analysis) | min. 98.0 % |
| Melting point | 115.0 to 119.0 °C |
| NMR | confirm to structure |
Properties (reference)
| Melting Point | 117 °C |
| Solubility in water | Insoluble |
| Degree of solubility in water | < 0.01 g/l |
| Solubility (soluble in) | dichloromethane |
| Solubility (insoluble in) | Methanol |
GHS
Related Laws:
Transport Information:
| H.S.code* | 2934.99-000 |
Application
Paliperidone Palmitate: A Prodrug of a Dopamine D2 and Serotonin 5-HT2 Receptors Antagonist, Paliperidone
Paliperidone palmitate is a long acting atypical antipsychotic agent. It is a prodrug that is metabolized by esterases to its active form paliperidone (9-hydroxyrisperidone) [P1897]. The active form paliperidone is a dopamine type 2 (D2) and serotonin type 2 (5-HT2) receptors antagonist, and the major active metabolite of the atypical antipsychotic risperidone [R0087]. (The product is for research purpose only.)
References
- Paliperidone palmitate – review of the efficacy, safety and cost of a new second-generation depot antipsychotic medication
- Comparative Pharmacology of Risperidone and Paliperidone (a review)
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