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CAS RN: 168273-06-1 | Product Number: R0205
Rimonabant
×
Purity: >98.0%(HPLC)
Synonyms:
- 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
- SR 141716
Product Documents:
| Size | Unit Price | Same Day | 2-3 Business Days | Other Lead Time |
Shipping Information
|
|---|---|---|---|---|---|
| 25MG |
$229.00
|
27 | 18 | Contact Us | |
| 100MG |
$684.00
|
0 | 14 | Contact Us |
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to order our products. The above prices do not include freight cost, customs, and other charges to the destination.
* The storage conditions are subject to change without notice.
| Product Number | R0205 |
Purity / Analysis Method 
|
>98.0%(HPLC) |
| Molecular Formula / Molecular Weight | C__2__2H__2__1Cl__3N__4O = 463.79 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature
|
Frozen (-20°C) |
| Store Under Inert Gas | Store under inert gas |
| Condition to Avoid | Air Sensitive,Heat Sensitive |
| CAS RN | 168273-06-1 |
| Reaxys Registry Number | 7231571 |
| PubChem Substance ID | 468592783 |
| MDL Number | MFCD04034714 |
Specifications
| Appearance | White to Almost white powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| NMR | confirm to structure |
Properties (reference)
GHS
| Pictogram |
|
| Signal Word | Warning |
| Hazard Statements | H361 : Suspected of damaging fertility or the unborn child. H371 : May cause damage to organs. H373 : May cause damage to organs through prolonged or repeated exposure. |
| Precautionary Statements | P501 : Dispose of contents/ container to an approved waste disposal plant. P260 : Do not breathe dust. P270 : Do not eat, drink or smoke when using this product. P202 : Do not handle until all safety precautions have been read and understood. P201 : Obtain special instructions before use. P264 : Wash skin thoroughly after handling. P280 : Wear protective gloves/ protective clothing/ eye protection/ face protection. P308 + P311 : IF exposed or concerned: Call a POISON CENTER/doctor. P405 : Store locked up. |
Related Laws:
| RTECS# | UQ6279632 |
Transport Information:
| H.S.code* | 2933.39-000 |
Application
Rimonabant: A Dual Inhibitor of Acyl CoA (cholesterol acyltransferase: ACAT) -1 and 2
Rimonabant and its hydrochloride [R0293] are also dual inhibitors of acyl-CoA (ACAT) 1 and 2, which catalyzes the intracellular synthesis of cholesteryl esters. (The product is for research use only.)
Reference
- Rimonabant is a dual inhibitor of acyl CoA:cholesterol acyltransferases 1 and 2
- Selective inhibition of sucrose and ethanol intake by SR 141716, an antagonist of central cannabinoid (CB1) receptors
- Keynote review: Medicinal chemistry strategies to CB1 cannabinoid receptor antagonists
- The psychiatric side-effects of rimonabant
- Development and validation of a high-performance liquid chromatographic method for bioanalytical application with rimonabant
Application
Rimonabant: A Selective Cannabinoid-1 Receptor (CB1) Antagonist.
Rimonabant (SR141716) is a selective cannabinoid-1 receptor (CB1) antagonist. CB1 is a G protein-coupled cannabinoid receptor that are found in the nervous system, and the body uses it to control food intake. It has been reported that rimonabant can help mammals to reduce food intake and to lose weight by blocking CB1 receptors. In clinical, rimonabant was withdrawn in 2008 due to serious psychiatric side effects. (The product is for research purpose only.)
References
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