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Risperidone
(CAS RN:106266-06-2 Product Number:R0087)

Structure

Risperidone
Synonym 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one

General Information

Product Number R0087

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Purity/Analysis Method >98.0%(HPLC)(T)
Storage Temperature
M.F. / M.W. C23H27FN4O2=410.49
CAS RN 106266-06-2
Related CAS RN
MDL Number MFCD00274576
Packaging and Container
  • Product Details
  • Safety & Regulations

Specification

Purity(HPLC) min. 98.0 area%
Purity(Nonaqueous Titration) min. 98.0 %
Melting point 170.0 to 174.0 deg-C

References

Reaxys-RN 4891881
PubChem SID 125307687
Merck Index(14) 8233
RTECS# UV1164800

GHS

Pictogram
Signal Word Danger
Hazard Statements
  • H301
  • :Toxic if swallowed.
Precautionary Statements
  • P264
  • :Wash hands and face thoroughly after handling.
  • P270
  • :Do not eat, drink or smoke when using this product.
  • P301+P310+P330
  • :IF SWALLOWED: Immediately call a POISON CENTER or doctor. Rinse mouth.
  • P405
  • :Store locked up.
  • P501
  • :Dispose of contents/container through a waste management company authorized by the local government.

Transport Information

UN Number 2811
Class 6.1
Packing Group III
HS Number 2934999090

Application

Risperidone: A Dopamine D2 and Serotonin 5-HT2 Receptors Antagonist

Risperidone, a benzisoxazole derivative, acts as a dopamine type 2 (D2) and serotonin type 2 (5-HT2) receptors antagonist. In addition, risperidone has affinity for α1- and α2-adrenergic, and H1 histaminergic receptors. While, risperidone has low to moderate affinity for the serotonin 5-HT1C, 5-HT1D and 5-HT1A receptors, week affinity for the dopamine D1 and haloperidol-sensitive sigma binding site, and no affinity for cholinergic muscarinic or β1 and β2 adrenergic receptors. Its major active metabolite is paliperidone (9-hydroxyrisperidone) [P1897]. Risperidone is used as a long acting antipsychotic agent with relatively few side effects. (The product is for research purpose only.)

References

PubMed Literature

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