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CAS RN: 29868-97-1 | Product Number: P2457
Pirenzepine Dihydrochloride
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Purity: >98.0%(T)(HPLC)
Synonyms:
- 5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Dihydrochloride
Product Documents:
| Size | Unit Price | Philadelphia, PA | Portland, OR | Japan* | Quantity |
|---|---|---|---|---|---|
| 200MG |
$42.00
|
2 | Contact Us | 5 |
|
| 1G |
$165.00
|
Contact Us | Contact Us | 4 |
|
* Items in stock locally ship in 1-2 business days. Items from Japan stock are able to ship from a US warehouse within 2 weeks. Please contact TCI for lead times on items not in stock. Excludes regulated items and items that ship on ice.
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*TCI frequently reviews storage conditions to optimize them. Please note that the latest information on the storage temperature for the products is described on our website.
| Product Number | P2457 |
Purity / Analysis Method 
|
>98.0%(T)(HPLC) |
| Molecular Formula / Molecular Weight | C__1__9H__2__1N__5O__2·2HCl = 424.33 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature
|
Room Temperature (Recommended in a cool and dark place, <15°C) |
| Packaging and Container
|
200MG-Glass Bottle with Plastic Insert (View image) |
| CAS RN | 29868-97-1 |
| Related CAS RN
|
28797-61-7 |
| Reaxys Registry Number | 4732388 |
| PubChem Substance ID | 468592608 |
| Merck Index (14) | 7491 |
| MDL Number | MFCD00055214 |
Specifications
| Appearance | White to Yellow to Orange powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| Purity(Argentometric Titration) | min. 98.0 %(calcd.on anh.substance) |
| Water | max. 4.9 % |
Properties (reference)
| Melting Point | 270 °C(dec.) |
| Solubility in water | Soluble |
| Solubility (slightly sol. in) | Methanol |
| Solubility (insoluble in) | Ether |
GHS
Related Laws:
| RTECS# | UU7883000 |
Transport Information:
| HS Number | 2933.99.7500 |
Application
Pirenzepine Dihydrochloride: A M1 Receptor Selective Antagonist
Pirenzepine dihydrochloride is a M1 receptor selective antagonist and a “selective” anti-ulcer agent. Unlike classic anticholinergic agents, pirenzepine inhibits gastric acid secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular and urinary functions. (The product is for research purpose only.)
References
- Pirenzepine. A review of its pharmacodynamic and pharmacokinetic properties and therapeutic efficacy in peptic ulcer disease and other allied diseases
- High performance liquid chromatographic determination of pirenzepine dihydrochloride in its pharmaceutical formulation
- Pirenzepine dihydrochloride (a review on the chemical detection method and pharmacology of it)
- HPLC determination of pirenzepine dihydrochloride in rabbit aqueous humor
Product Articles
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Specifications
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