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CAS RN: 85118-33-8 | 產品號碼: G0405
Gaboxadol Hydrochloride
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| 產品號碼 | G0405 |
純度/分析方法 
|
>98.0%(HPLC) |
| 分子式 / 分子量 | C__6H__8N__2O__2·HCl = 176.60 |
| 外觀與形狀（20°C） | Solid |
| 儲存條件
|
Room Temperature (Recommended in a cool and dark place, <15°C) |
| 包裝和容器
|
25MG-Glass Bottle with Plastic Insert （閲覽圖片） |
| CAS RN | 85118-33-8 |
| 相關CAS RN
|
64603-91-4 |
| Reaxys-RN | 6534899 |
| PubChem Substance ID | 253659629 |
| Merck Index(14) | 4321 |
| MDL編號 | MFCD00055180 |
產品規格
| Appearance | White to Almost white powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| Elemental analysis(Nitrogen) | 15.40 to 16.30 % |
性質
| 熔點 | 236 °C |
GHS
相關法規
| RTECS # | NY3398000 |
運輸資料
| HS編碼* | 2934.99-000 |
Application
Gaboxadol Hydrochloride: A γ-Aminobutyric Acid Subtype A (GABAA) Receptor Agonist
Gaboxadol hydrochloride, also known as THIP, is a direct-acting γ-aminobutyric acid subtype A (GABAA) receptor agonist. GABAA receptor is widely considered to be an important target for most clinically effective sedative-hypnotic compounds. However, the clinical development program for gaboxadol was discontinued in 2007. (The product is for research purpose only.)
References
- Pharmacological characterization of a novel cell line expressing human α4β3δ GABAA receptors
- GABAA receptor α4 subunits mediate extrasynaptic inhibition in thalamus and dentate gyrus and the action of gaboxadol
- An extrasynaptic GABAA receptor mediates tonic inhibition in thalamic VB neurons
- Gaboxadol - a new awakening in sleep(a review)
- GABAA agonists and partial agonists: THIP (Gaboxadol) as a non-opioid analgesic and a novel type of hypnotic(a review)
- Development and validation of a selective and sensitive bioanalytical procedure for the quantitative determination of gaboxadol in human plasma employing mixed mode solid phase extraction and hydrophilic interaction liquid chromatography with tandem mass spectroscopic detection
PubMed Literature
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