Maximum quantity allowed is 999
Please select the quantity
CAS RN: 199739-10-1 | Product Number: P2967
Paliperidone Palmitate
×
![]()
×
Purity: >98.0%(T)(HPLC)
Synonyms:
- 9-Hydroxyrisperidone Palmitate
- 3-[2-[4-(6-Fluoro-1,2-benzoxazol-3-yl)-1-piperidinyl]ethyl]-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl Palmitate
Product Documents:
| Size | Unit Price | Shanghai | Tianjin | Japan* |
|---|---|---|---|---|
| 100MG |
¥190.00
|
9 | Contact Us | 8 |
| 1G |
¥690.00
|
5 | Contact Us | 16 |
* For order or inquiry, please contact
Our Authorized Distributors.
*TCI frequently reviews storage conditions to optimize them. Please note that the latest information on the storage temperature for the products is described on our website.
* To send your quote request for bulk quantities, please click on the "Request Bulk Quote" button. Please note that we cannot offer bulk quantities for some products.
| Product Number | P2967 |
Purity / Analysis Method 
|
>98.0%(T)(HPLC) |
| Molecular Formula / Molecular Weight | C__3__9H__5__7FN__4O__4 = 664.91 |
| Physical State (20 deg.C) | Solid |
| Storage Temperature
|
Refrigerated (0-10°C) |
| Store Under Inert Gas | Store under inert gas |
| Condition to Avoid | Air Sensitive,Heat Sensitive |
| Packaging and Container
|
100MG-Glass Bottle with Plastic Insert (View image), 1G-Glass Bottle with Plastic Insert (View image) |
| CAS RN | 199739-10-1 |
| Reaxys Registry Number | 15026585 |
| MDL Number | MFCD24386477 |
Specifications
| Appearance | White to Light yellow powder to crystal |
| Purity(HPLC) | min. 98.0 area% |
| Purity(Volumetric Analysis) | min. 98.0 % |
| Melting point | 115.0 to 119.0 °C |
| NMR | confirm to structure |
Properties (reference)
| Melting Point | 117 °C |
| Solubility in water | Insoluble |
| Degree of solubility in water | < 0.01 g/l |
| Solubility (soluble in) | dichloromethane |
| Solubility (insoluble in) | Methanol |
GHS
Related Laws:
Transport Information:
| Customs Control Conditions (Q) |
Application
Paliperidone Palmitate: A Prodrug of a Dopamine D2 and Serotonin 5-HT2 Receptors Antagonist, Paliperidone
Paliperidone palmitate is a long acting atypical antipsychotic agent. It is a prodrug that is metabolized by esterases to its active form paliperidone (9-hydroxyrisperidone) [P1897]. The active form paliperidone is a dopamine type 2 (D2) and serotonin type 2 (5-HT2) receptors antagonist, and the major active metabolite of the atypical antipsychotic risperidone [R0087]. (The product is for research purpose only.)
References
- Paliperidone palmitate – review of the efficacy, safety and cost of a new second-generation depot antipsychotic medication
- Comparative Pharmacology of Risperidone and Paliperidone (a review)
Product Documents (Note: Some products will not have analytical charts available.)
Safety Data Sheet (SDS)
Please select Language.
The requested SDS is not available.
Please Contact Us for more information.
Specifications
C of A & Other Certificates
Please enter Lot Number
Incorrect Lot Number. Please input only the 4-5 alphanumeric characters before the hyphen.
Sample C of A
This is a sample C of A and may not represent a recently manufactured lot of the product.
A sample C of A for this product is not available at this time.
Analytical Charts
Please enter Lot Number
Incorrect Lot Number. Please input only the 4-5 alphanumeric characters before the hyphen.
The requested analytical chart is not available. Sorry for the inconvenience.